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They suppress activation of ?1-receptors without a concomitant enhancement of norepinephrine release. ?1-Blockers may be used in hypertension.
The initiation of an epileptic attack involves “pacemaker” cells; these differ from other nerve cells in their unstable resting membrane potential, i. e. , a depolarizing membrane current persists after the action potential terminates. Therapeutic interventions aim to stabilize neuronal resting potential and, hence, to lower excitability. |
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